COMPOUNDS AS MODULATING AGENTS OF STEROID RECEPTORS AND METHODS Russian patent published in 2002 - IPC

Abstract RU 2191774 C2

FIELD: organic chemistry, pharmacy. SUBSTANCE: invention relates to nonsteroid compounds that present highly affinitive modulating agents of steroid receptors. Invention describes also pharmaceutical composition comprising such compounds. Invention discloses intermediate compounds useful for preparing these compounds and methods of synthesis of compounds as modulating agents of steroid receptors. Invention can be used in medicine as therapeutic agent as modulating agent (i. e. agonist and antagonist) of steroid receptors (for example, receptor of progesterone, androgen, estrogen and others). EFFECT: improved method of preparing and synthesis, valuable medicinal properties of agents. 49 cl, 9 tbl, 362 ex

Similar patents RU2191774C2

Title Year Author Number
DERIVATIVES OF 8-PYRIDONO[5,6-G]QUINOLINE, PHARMACEUTICAL COMPOSITION AND METHOD FOR CONTROL WITH THEIR USING 1997
  • Ehdvardz Dzhejms P.
  • Khiguchi Robert
  • Dzhons Todd
RU2214412C2
Axl INHIBITORS APPLICABLE IN COMBINATION THERAPY FOR PREVENTING, RELIEVING OR TREATING METASTATIC CANCER 2010
  • Khotosi Jasumiti
  • Kholland Sasha
  • Pajjan Donal'D Dzh.
RU2555326C2
TETRAHYDROACRIDINE DERIVATIVES, PROCESSES FOR PREPARATION THEREOF (VARIANTS), TETRAHYDROACRIDINONE DERIVATIVES, DIHYDROBENZOXAROLE DERIVATIVE AND PHARMACEUTIC COMPOSITION HAVING EFFECT OF EASING OR ELIMINATING MEMORY DYSFUNCTION 1992
  • Gregori Majkl Shatski[Us]
  • Kevin Dzhejms Kaples[Us]
  • Dzhon Dik Tomer[Us]
RU2083564C1
MODULATORS OF ATP-BINDING TRANSPORTERS 2010
  • Shet Urvi
  • Fehnning Lev T. D.
  • Numa Mekhdi
  • Binch Khehjli
  • Kharli Dennis Dzhejms
  • Chzhou Tszinlan'
  • Adida Rua Sara S.
  • Khejzlvud Anna R.
  • Silina Alina
  • Vairagoundar Radzhendran
  • Van Gur Frederik F.
  • Grotenkhejs Peter Diderik Jan
  • Botfild Martin K.
RU2552353C2
TETRAHYDROQUINOLINE DERIVATIVES 2002
  • Van Straten Nikol' Korin Rene
  • Van Someren Rudol'F Gejsbertus
  • Shul'Ts Jurgen
RU2347570C2
MODULATORS OF ATP-BINDING CARTRIDGE TRANSPORTERS 2005
  • Adida Rua Sara S.
  • Khejzlvud Anna R.
  • Grotenkhejs Peter D.,J.
  • Van Gur Frederik F.
  • Singkh Ashvani K.
  • Chzhou Tszinlan'
  • Makkartni Dzhejson
RU2528046C2
BICYCLIC PYRIDINES AND ANALOGUES AS SIRTUIN MODULATORS 2010
  • Ng Pui Ji
  • Blum Charl'Z
  • Makferson Loren
  • Perni Robert B.
  • Vu Chi B.
  • Akhmed Mokhammed Makhmud
  • Dish Dzheremi S.
RU2550821C2
HETEROCYCLIC COMPOUNDS AND THEIR APPLICATION AS GLYCOGEN SYNTHASE KINASE-3 INHIBITORS 2011
  • Terner Shon Kolm
  • Mak Khelmut
  • Bakker Margareta Khenrika Mariya
  • Van Galen Marsel
  • Khoft Karolin
  • Khornberger Vilfrid
RU2623427C2
METHODS AND COMPOSITIONS FOR GROWTH STIMULATION OF NEURITIS 1996
  • Armistid Dehvid M.
RU2197240C2
MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS 2005
  • Adida Rua Sara S
  • Khejzlvud Anna R
  • Grotenkhejs Peter D J
  • Van Gur Frederik F
  • Singkh Ashvani K
  • Chzhou Tszinlan'
  • Makkartni Dzhejson
RU2556984C2

RU 2 191 774 C2

Authors

Dzhounz Todd K.

Goldman Mark E.

Pulej Sharlotte L. F.

Vinn Dehvid T.

Ehdvardz Dzhejms E.

Vest Sara Dzh.

Tegli Kristofer M.

Zhi Lin

Khamann Lorens G.

Farmer Ljuk Dzh.

Dehvis Robert Dzh.

Dates

2002-10-27Published

1995-12-13Filed