FIELD: organic chemistry, pharmacy. SUBSTANCE: invention relates to new derivatives of 2-aminopyridine of the general formula (I): wherein A means radical of the formula: wherein R1, R2, R3 mean hydrogen, halogen atom, hydroxyl, alkyl or alkoxy-group, and other groups; or radical of the formula: wherein R8 means hydrogen atom; X means radical -(CH2)m-Q; m is a whole number from 0 to 6; Y means alkyl, alkenyl, alkynyl chain and others; R10 means hydrogen atom or alkyl, or to their salts. Compounds of the formula (I) elicit inhibitory effect with respect to activity of NO-synthases and can be used in medicine. EFFECT: valuable medicinal properties of compounds. 11 cl, 36 ex
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Authors
Dates
2004-04-10—Published
1999-07-05—Filed