FIELD: organic chemistry, medicine, oncology.
SUBSTANCE: invention relates to new derivatives of 2-arylimino-2,3-dihydrothiazoles of the general formula (I): wherein radical values R1, R2, R3 and R4 are given in the claim invention. New compounds are useful in treatment of pathological states or diseases wherein one or some somatostatin receptors are implicated, for example, acromegaly, hypophysis adenomas or gastroenteropancreatic endocrine tumors with carcinoid syndrome and gastroenteric bleedings.
EFFECT: improved preparing method, valuable medicinal properties of compounds and compositions.
14 cl, 2825 ex
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Authors
Dates
2005-12-20—Published
2000-07-21—Filed