2-ARYLIMINO-2,3-DIHYDROTHIAZOLES, METHODS FOR THEIR PREPARING AND PHARMACEUTICAL COMPOSITION COMPRISING THEREOF Russian patent published in 2005 - IPC

Abstract RU 2266287 C2

FIELD: organic chemistry, medicine, oncology.

SUBSTANCE: invention relates to new derivatives of 2-arylimino-2,3-dihydrothiazoles of the general formula (I): wherein radical values R1, R2, R3 and R4 are given in the claim invention. New compounds are useful in treatment of pathological states or diseases wherein one or some somatostatin receptors are implicated, for example, acromegaly, hypophysis adenomas or gastroenteropancreatic endocrine tumors with carcinoid syndrome and gastroenteric bleedings.

EFFECT: improved preparing method, valuable medicinal properties of compounds and compositions.

14 cl, 2825 ex

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RU 2 266 287 C2

Authors

Muane Kristof

Sakjur Karol'

Tjur'O Kristof

Dates

2005-12-20Published

2000-07-21Filed