FIELD: organic chemistry, medicine, pharmacy.
SUBSTANCE: invention relates to new derivatives of 3-hydroxypiperidine of the general formula (I): 
wherein R means (a): -C(O)(CH2)nC(O)OH; (b): 
wherein R1 means -N(R2)(R3); each R2 and R3 means hydrogen atom, lower alkyl or cyclic tertiary amine; (c): -P(O)(OH)2 or (d): -C(O)(CH2)n and -NHC(O)(CH2)nN(R2)(R3) wherein n means a whole number 1-4. Indicated compounds can be used as prodrugs in preparing medicinal agents used in treatment of diseases associated with blocking agents for receptors of subtype NMDA.
EFFECT: valuable medicinal properties of compounds and composition.
10 cl, 1 tbl, 20 ex
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