PHARMACEUTICAL COMPOSITION WITH STABLE SUSTAINED-RELEASE FOR PARENTERAL ADMINISTRATION OF BIOLOGICALLY ACTIVE HYDROPHILIC SUBSTANCES Russian patent published in 2006 - IPC A61K9/107 

Abstract RU 2272615 C2

FIELD: medicine, chemical-pharmaceutical industry.

SUBSTANCE: invention relates to a stable, biologically compatible and good tolerated microemulsion of type water-in-oil designated for the parenteral administration of biologically active hydrophilic compounds or converting to such compounds as result of corresponding derivatization and providing the stable and sustained-release of active substances comprising in it. The claimed microemulsion shows low toxicity, high tolerance and provides the prolonged effect of active substance for a long time.

EFFECT: improved and valuable properties of compositions.

16 cl, 4 dwg, 6 tbl, 15 ex

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RU 2 272 615 C2

Authors

Autuori Franchesko

B'Jankini Karlo

Bottoni Dzhuzeppe

Leoni Flavio

Maskan'I Paolo

Montsani Val'Men

Pikkolo Oreste

Dates

2006-03-27Published

2001-05-23Filed