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2 286 340

(13)

(51)

IPC

C07D239/96(2006-01-01)

C07D239/93(2006-01-01)

C07D239/94(2006-01-01)

C07D401/12(2006-01-01)

C07D239/78(2006-01-01)

C07D253/08(2006-01-01)

A61K31/517(2006-01-01)

A61K31/53(2006-01-01)

A61K31/519(2006-01-01)

A61K31/549(2006-01-01)

A61P43/00(2006-01-01)

A61P29/00(2006-01-01)

A61P19/02(2006-01-01)

A61P1/04(2006-01-01)

(21) (22)

Application

2003104821/04, 2001-08-15

(24)

Start date

2001-08-15

(22)

Actual filing date

2001-08-15

(45)

Published

2006-10-27

(72)

Inventor

Makino SingoOkuzumi TatsujaJosimura TosikhikoSatake JukoSuzuki NobujasuIzava KhirojukiSagi KazujukiTiba AkiraNakanisi EidziMurata MasakhiroTsudzi Takasi

(73)

Holder

Adzinomoto Ko., Ink.

NOVEL DERIVATIVES OF PHENYLALANINE Russian patent published in 2006 - IPC C07D239/96 C07D239/93 C07D239/94 C07D401/12 C07D239/78 C07D253/08 A61K31/517 A61K31/53 A61K31/519 A61K31/549 A61P43/00 A61P29/00 A61P19/02 A61P1/04

Abstract RU 2286340 C2

FIELD: organic chemistry, amino acids.

SUBSTANCE: invention proposes the novel derivatives of phenylalanine of the formula (I) and (II) possessing with antagonistic activity with respect to α4-integrin. Derivatives of phenylalanine are used as therapeutic agents in different diseases associated with α4-integrin.

EFFECT: valuable medicinal properties of compounds.

37 cl, 30 tbl, 215 ex

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RU 2 286 340 C2

Authors

Makino Singo

Okuzumi Tatsuja

Josimura Tosikhiko

Satake Juko

Suzuki Nobujasu

Izava Khirojuki

Sagi Kazujuki

Tiba Akira

Nakanisi Eidzi

Murata Masakhiro

Tsudzi Takasi

Dates

2006-10-27—Published

2001-08-15—Filed