DERIVATIVES OF 4-PIPERIDINYLALKYLAMINE AND PHARMACEUTICAL COMPOSITION POSSESSING ANTAGONISTIC AFFECT ON MUSCARINIC RECEPTOR Russian patent published in 2007 - IPC C07D211/62 C07D211/96 C07D401/12 C07D405/06 C07D407/12 C07D409/06 C07D409/12 C07D413/06 C07D413/12 C07D413/14 A61K31/455 A61K31/495 A61P1/00 A61P11/00 

Abstract RU 2300524 C2

FIELD: organic chemistry, medicine, pharmacy.

SUBSTANCE: invention describes novel compounds of the general formula (I) wherein p, R1, R2, R3 and A are determined in the invention description, their individual isomers and their pharmaceutically acceptable salts. Proposed compounds possess antagonistic effect with respect to muscarinic receptors that allows their using in treatment and prophylaxis of diseases yielding to treatment with muscarinic receptor antagonist. Also, invention describes a pharmaceutical composition containing these compounds.

EFFECT: valuable medicinal properties of compounds and pharmaceutical composition.

23 cl, 22 ex

Similar patents RU2300524C2

Title Year Author Number
SUBSTITUTED 1-AMINOALKYL LACTAMS, PHARMACEUTICAL COMPOSITION BASED ON THEREOF AND METHOD FOR THEIR PREPARING 2001
  • Madera Ann Marie
  • Stabler Rassell Stiven
  • Uejkert Robert Dzhejms
RU2243222C2
DERIVATIVES OF AMINOTETRALINE AS MUSCARINIC RECEPTOR ANTAGONIST 2002
  • Madera Ann Mari
  • Uehjkert Robert Dzhejms
RU2311408C2
DERIVATIVES OF 1,2,3,4-TETRAHYDRONAPHTHALENE, METHODS OF THEIR SYNTHESIS, PHARMACEUTICAL COMPOSITION BASED ON THEREOF AND METHOD OF TREATMENT 1998
  • Berg Stefan
  • Linderberg Mats
  • Ross Svante
  • Torberg Set-Olov
  • Ul'Ff Bengt
RU2194696C2
NOVEL PHOSPHATE COMPOUNDS, SYNTHESIS METHOD THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME 2014
  • Le-Tiran Arno
  • Le-Digarer Terri
  • Stark Zherom-Benua
  • Anlen Zhan-Mishel
  • Gijuzi Anne-Fransua
  • De-Nantej Gijom
  • Zhenes Olive
  • Dejvidson Dzhejms Eduard Pol
  • Marri Dzhejms Bruk
  • Chen Itszen
RU2617682C2
NEW INDOLIZINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM 2013
  • Le-Digare Terri
  • Kasara Patrik
  • Stark Zherom-Benua
  • Anlen Zhan-Mishel
  • Dejvidson Dzhejms Eduard Pol
  • Marri Dzhejms Bruk
  • Grem Kristofer Dzhon
  • Chen Itszen
  • Zhenes Olive
  • Khikman Dzhon
  • Depil Stefan
  • Le-Tiran Arno
  • Niergesh Miklosh
  • De-Nantej Gijom
RU2646223C2
INDAZOL DERIVATIVES AS CRF ANTAGONISTS 2003
  • Kurnojer Richard Leo
  • Lokhed Dejvid Garrett
  • O`Jang Kund
RU2341518C2
STIMULATING AGENTS OF GROWTH HORMONE SECRETION 1996
  • Filip A. Karpino
  • Pol A. Dasil'Va Dzhardin
  • Brjus A. Lefker
  • Dzhon A. Rehgehn
RU2172742C2
1-[M-CARBOXAMIDO(HETERO)ARYL-METHYL]-HETEROCYCLYL-CARBOXAMIDE DERIVATIVES 2013
  • Fretts Khajnts
  • Gude Markus
  • Gerri Filipp
  • Kimmerlen Terri
  • Leembre Fransua
  • Pfajfer Tomas
  • Valdener Anya
RU2644761C2
AMINOPYRIDINE-CONTAINING SPLEEN TYROSINE KINASE (SYK) INHIBITORS 2012
RU2612217C2
PYRIMIDINE AMIDE COMPOUNDS AS PGDS INHIBITORS 2006
  • Oldous S'Juzan S.
  • Tszjan' Dzhon Tszytsi
  • Lu Tszin'Tsi
  • Ma Ljan
  • Mu Lan'
  • Manson Khehrri Rendall
  • Sejbol Dzheffri Stefen
  • Tkhurajratnam Sukantkhini
  • Vandjuzen Kristofer Loren
RU2420519C2

RU 2 300 524 C2

Authors

Broterton-Plejss Kristine Eh.

Madera Ann Mari

Uehjkert Robert Dzhejms

Dates

2007-06-10Published

2002-11-25Filed