AZAINDOLEOXOACETIC DERIVATIVES OF PIPERAZINE AND PHARMACEUTICAL COMPOSITION BASED ON THEREOF Russian patent published in 2007 - IPC C07D401/14 C07D403/14 A61K31/496 A61P31/18 

Abstract RU 2303038 C2

FIELD: organic chemistry, medicine, pharmacy.

SUBSTANCE: invention relates to azaindoleoxoacetic derivatives of piperazine of the general formula (I): wherein Q is chosen from the group consisting of the following compounds: ; -W- represents compound of the formula: . Proposed compounds possess antiviral activity both in separate using and in combination with other antiviral, anti-infectious agents, immunomodulating agents or inhibitors HIV entering. Also, invention describes a pharmaceutical composition based on compounds of the formula (I).

EFFECT: valuable medicinal properties of compounds and pharmaceutical composition.

55 cl, 10 tbl, 169 ex

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RU 2 303 038 C2

Authors

Vang Tao

Zkhang Zkhongksing

Minvell Nikolas A.

Kehdou Dzhon F.

Jin Zkhivej

Dates

2007-07-20Published

2002-01-02Filed