NON-NUCLEOSIDE REVERSE TRANCRIPTASE INHIBITORS, USES THEREOF, PHARMACEUTICAL COMPOSITION FOR HIV INHIBITION Russian patent published in 2007 - IPC C07D231/20 C07D403/06 C07D401/06 C07D409/06 A61K31/4155 A61P31/18

Abstract RU 2305680 C2

FIELD: organic chemistry.

SUBSTANCE: invention relates to new pyrasole derivatives of formula I wherein R⁵ represents phenyl or heteroaryl ring of formulae IIIa-IIIh meanings of the rest substituents are as defined in specification. Also disclosed are pharmaceutical composition based on said derivatives of formula I and uses thereof.

EFFECT: new biologically active compounds and pharmaceutical compositions based on the same for HIV inhibition.

13 cl, 54 ex, 2 tbl

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RU 2 305 680 C2

Authors

Dann Dzhejms Patrik

Khogg Dzhoan Kheder

Mirzadegan Taranekh

Svolou Stiven

Dates

2007-09-10—Published

2004-02-17—Filed