FIELD: organic chemistry, medicine.
SUBSTANCE: invention relates to compounds of formula I 
, wherein G is carbon or nitrogen atom; A is i) phenyl substituted with any from -COOH, -CONH2, COOCH3, -CN, -NH2 or -COCH3; ii) naphthyl, benzophuranyl, and quinolinyl; and iii) formulae 
, 
, 
.
Compounds of present invention are useful in particular in pain treatment.
EFFECT: new agents for pain treatment.
58 ex
| Title | Year | Author | Number |
|---|---|---|---|
| DERIVATIVES OF PIPERAZINE AND PIPERIDINE AND PHARMACEUTICAL COMPOSITION | 1996 |
|
RU2194702C2 |
| METHOD FOR SYNTHESIS OF 3-ARYLINDAN-1-ONES BY REACTION OF SUPER-ELECTROPHILIC AROMATIC SUBSTITUTION OF CINNAMIC NITRILES | 2020 |
|
RU2768714C2 |
| 1-METHYLCARBAPENEM DERIVATIVES, METHOD OF PREPARING THEREOF, PHARMACEUTICAL COMPOSITION BASED THEREON, AND METHOD OF ANTIBACTERIAL EFFECT | 1996 |
|
RU2160737C2 |
| VITAMIN D ANALOGS, METHODS OF THEIR SYNTHESIS, PHARMACEUTICAL COMPOSITION | 1994 |
|
RU2153491C2 |
| 4-PIPERAZINYL-(8-QUINOLINYL)-METHYL)-BENZAMIDES, PHARMACEUTICAL COMPOSITION AND METHOD FOR PAIN TREATMENT | 2000 |
|
RU2260006C2 |
| METHOD FOR IMPROVEMENT OF STABILITY OF SWEET TASTE INTENSIFIERS AND COMPOSITION CONTAINING STABILISED SWEET TASTE INTENSIFIER | 2011 |
|
RU2576451C2 |
| BI-ARYL-META-PYRIMIDINE KINASE INHIBITORS | 2006 |
|
RU2597364C2 |
| BI-ARYL-META-PYRIMIDINE KINASE INHIBITORS | 2006 |
|
RU2589878C2 |
| NOVEL PYRROLE DERIVATIVE HAVING AS SUBSTITUTES UREIDE GROUP, AMINOCARBONYL GROUP AND BICYCLIC GROUP, OPTIONALLY SUBSTITUTED | 2009 |
|
RU2500669C2 |
| DERIVATIVES OF CHINOLINESULPHONAMIDES AND THEIR APPLICATION FOR MODULATION OF PKM2 ACTIVITY | 2010 |
|
RU2561132C2 |
