SUBSTITUTED DIKETOPIPERAZINS AND THEIR APPLICATION AS OXYTOCENE ANTAGONISTS Russian patent published in 2009 - IPC C07D413/14 A61K31/496 A61P15/06 

Abstract RU 2343152 C2

FIELD: chemistry.

SUBSTANCE: in substituted diketopiperazins of general formula I R1 represents 2-indanyl, R2 represents 1-methylpropyl, R3 represents 2-methyl-1,3-oxazol-4-yl and R4 and R5 together with nitrogen atom to which they are bound, represent morpholyno.

EFFECT: antagonistic effect on oxytocene receptor, possibility of their application in medicine.

11 cl, 3 ex

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RU 2 343 152 C2

Authors

Liddl Dzhon

Dates

2009-01-10Published

2004-06-22Filed