FIELD: chemistry.
SUBSTANCE: in substituted diketopiperazins of general formula I R1 represents 2-indanyl, R2 represents 1-methylpropyl, R3 represents 2-methyl-1,3-oxazol-4-yl and R4 and R5 together with nitrogen atom to which they are bound, represent morpholyno.
EFFECT: antagonistic effect on oxytocene receptor, possibility of their application in medicine.
11 cl, 3 ex
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Authors
Dates
2009-01-10—Published
2004-06-22—Filed