STABLE MODIFICATIONS OF TEGASEROD HYDROMALEATE Russian patent published in 2009 - IPC C07D209/14 A61K31/404 A61P1/04 

Abstract RU 2349585 C2

FIELD: chemistry.

SUBSTANCE: present invention pertains to crystal forms of tegaserod hydromaleate, their use in pharmaceutical compositions, suitable for treating irritated bowel syndrome, gastroesophageal reflux disease, functional dyspepsia, chronic constipation or diarrhea. The invention also relates to production of these modifications.

EFFECT: obtaining new stable crystal forms of tegaserod hydromaleate, distinguished by stability when heated and in the presence of water.

10 cl, 9 ex, 3 tbl, 5 dwg

Similar patents RU2349585C2

Title Year Author Number
NEW COMPOSITION FOR ORAL ADMINISTRATION 1999
  • De-Bruejn Karel
  • Ehngel' Gjunter
  • Pfannkukhe Khans-Jurgen
  • Tevissen Mikhaehl'
  • Vitzleng Kristian
  • Tsjuger Otmar
RU2260424C9
PHARMACEUTICAL COMPOSITIONS CONTAINING PARTIAL 5HTAGONIST 2002
  • Ober Zherom
  • Vitzling Kristian
RU2322978C2
2,6-SUBSTITUTED-4-MONOSUBSTITUTED AMINOPYRIMIDINES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS 2007
  • Stefani Dehvid
  • Kharris Kit Dzhon
  • Gillespi Timoti Alan
  • Gardner Charl'Z Dzh.
  • Agiar Zhuasi K.
RU2431631C2
PURIFIED PYRROLOQUINOLINYL-PYRROLIDINE-2,5-DIONE COMPOSITIONS AND METHODS OF OBTAINING AND APPLICATION THEREOF 2010
  • Rid Dehvid P.
  • Barns Nil R.
  • Kejn Dzhon K.
  • Li Kristofer A.
  • Chehn' Tszjan'-Se
  • Redmond Martin P.
RU2556205C2
TREATMENT OF DERMATOLOGICAL ALLERGIC STATES 2011
  • Choi-Sledeski Jong Mi
  • Fitch Nejl
  • Minnikh Anne
RU2521357C2
[4-(5-AMINOMETHYL-2-FLOUROPHENYL)-PYPERIDIN-1-YL]-(7- FLUORO-1-(2-METHOXYETHYL)-4-TRIFLUOROMETHOXY-1H-INDOL-3-YL]-METHANONE AS MAST CELL TRYPTASE INHIBITOR 2009
  • Choi-Sledeski Jong Mi
  • Choj Nakien
  • Poli Gregori Bernard
  • Shej Dzhon Dzh. Ml.
  • Shum Patrik Vai-Kvok
  • Sledeski Adam V.
RU2509766C2
ALKOXY-SUBSTITUTED BENZIMIDAZOLE COMPOUNDS, PHARMACEUTICAL PREPARATIONS COMPRISING THEREOF AND METHOD FOR THEIR USING 2000
  • Uittl Robert R.
  • Sanchilio Frederik D.
  • Stouehll Grehjson Uoker
  • Dzhenkins Duglas Dzhon
  • Uittol Linda
  • Mejer Glenn Alan
  • Fontana Stiven A.
RU2263673C2
4-PYPERAZINYL-BENZEN-SULFANYLINDOLES WITH AFFINITY TO 5-HT6 RECEPTOR 2003
  • Klark Robin Duglas
  • Kharris Ralf N'Ju Iii
  • Repke Dejvid Brjus
RU2324693C2
INDOLE DERIVATIVES AND PHYSIOLOGICALLY ACCEPTABLE SALTS AND SOLVATES THEREOF, METHODS OF PREPARING THEREOF, DRUG FOR TREATMENT OR PROPHYLAXES OF CLINICAL STATES FOR WHICH ADMINISTRATION OF 5-HT-LIKE RECEPTOR AGONIST, AND METHOD OF PREPARING THEREOF 1991
  • Alan Dunkan Robertson
  • Alan Piter Khill
  • Robert Charl'Z Glen
  • Grem Richard Martin
RU2160736C2
TETRAHYDRO-1H-PYRIDO[3,4-B]INDOLE ANTI-ESTROGENIC DRUGS 2016
  • Myles, David, C.
  • Kushner, Peter, J.
  • Harmon, Cyrus, L.
RU2745742C1

RU 2 349 585 C2

Authors

Pfeffer Zabine

Vittsling Kristian

Dates

2009-03-20Published

2004-07-23Filed