4-PYPERAZINYL-BENZEN-SULFANYLINDOLES WITH AFFINITY TO 5-HT6 RECEPTOR Russian patent published in 2008 - IPC C07D403/12 A61K31/496 A61P25/00 

Abstract RU 2324693 C2

FIELD: medicine; pharmacology.

SUBSTANCE: invention is related to 4-pyperazinyl-benzen-sulfanylindols with the general formula I , where: R1 and R2 each independently means hydrogen, halogen, alcoxy, R3 and R4 each independently means hydrogen, halogen, alkyl, n is equal to 0 to 4, R6 in each particular case means hydrogen or halogen, R7 and R8 each means hydrogen, R9 means hydrogen, alkyl, or individual isomer, racemic or non-racemic mixture of isomers or their pharmaceutically acceptable salt or solvate. The pharmaceutical compositions are described based on compound I.

EFFECT: compounds can be efficiently used in treatment of certain diseases of central nervous system.

14 cl, 1 tbl, 4 ex

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RU 2 324 693 C2

Authors

Klark Robin Duglas

Kharris Ralf N'Ju Iii

Repke Dejvid Brjus

Dates

2008-05-20Published

2003-10-13Filed