STABLE FORMULATION FROM PHENYLALANINE DERIVATIVES Russian patent published in 2009 - IPC A61K31/4965 A61K47/10 A61P35/04 

Abstract RU 2358736 C2

FIELD: medicine.

SUBSTANCE: invention refers to medical products and concerns pharmaceutical composition for treatment of the diseases associated with urokinase activator of plasminogen (u-PA) and/or with receptor of activator of urokinase plasminogen (u-PAR), containing: (i) amidino-, hydroxyamidino-, guanydino- and/or hydroxyguanydinophenylalanine derivative as an active material, (ii) mixed alcohol and polyol, and (iii) aqueous phase containing buffer solution. There is also disclosed stabilisation method of pharmaceutical composition.

EFFECT: physical and chemical stability.

25 cl, 6 dwg, 1 tbl, 9 ex

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RU 2 358 736 C2

Authors

Shmaliks Vol'Fgang

Bjurgle Markus

Kokh Klaus

Dates

2009-06-20Published

2005-09-20Filed