FIELD: chemistry.
SUBSTANCE: invention relates to new phosphates of nitrophenylpyrite and nitrophenylaziridine alcohols of general formula 
, where: X represents -CONH- in any accessible position of the ring; R is a lower C1-6alkyl; Y represents -N-aziridinyl in any accessible position of the ring, -N(CH2CH2W)2 or -N(CH2CHMeW)2, where W is independently chosen from halogen or -OSO2Me; Z represents NO2 or -SO2Me in any accessible position of the ring; and its pharmaceutically acceptable salts. The invention also pertains to a method of producing phosphates of formula (I) and formulae 
, 
and 
(particular cases of formula (I)), a method of anticancer treatment and a method of destroying hypoxic cells using formula (I) compounds, as well as to a pharmaceutical composition based on formula (I) compounds.
EFFECT: obtaining new compounds which can be used as targeted cytotoxic agents.
14 cl, 5 tbl, 4 dwg, 39 ex
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