FIELD: chemistry.
SUBSTANCE: new pyrrolotriazine derivatives of general formula (I) are described, where R1 is possibly substituted piperidinyl or piperazinyl; R2 is possibly substituted phenyl; R3 is hydrogen; X is -NH-; Y is -CH2-; as well as their pharmaceutically acceptable salts or steroisomers, and pharmaceutical compositions containing said compounds.
EFFECT: given compounds are kinase inhibitors and can be used in medicine, for example as anticancer agents.
9 cl, 267 ex, 2 dwg
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Authors
Dates
2009-11-20—Published
2004-12-23—Filed