FIELD: chemistry.
SUBSTANCE: invention relates to organic chemistry, and specifically to (2R)-2-{(1S)-6,7-dimethoxy-1-[2-(4-trifluoromethylphenyl)-ethyl]-3,4-dihydro-1H-isoquinolin-2-yl}-N-methyl-2-phenylacetamide or pharmaceutically acceptable salt thereof. The invention also relates to use and a pharmaceutical composition based on said compound with non-peptide antagonistic activity of human orexin receptors.
EFFECT: obtaining a novel compound and its salt, which can be used in medicine as a medicinal agent for preventing or treating diseases such as nutritional and sleep disorders.
11 cl, 3 tbl, 4 ex
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