PEPTIDES HAVING AGONISTIC ACTIVITY ON NEUROPEPTIDE-2 RECEPTOR (Y2R) Russian patent published in 2010 - IPC C07K14/575 C07K7/08 A61K38/22 A61K38/10 A61P5/48

Abstract RU 2383553 C2

FIELD: chemistry.

SUBSTANCE: invention relates to agonists of neuropeptide-2 receptor with formula (I): Y-R₁-R₂-X-R₃-R₄-R₅-R₆-R₇-R₈-R₉-R₁₀-R₁₁-R₁₂-R₁₃-R₁₄-NH₂(l), as well as their pharmaceutically acceptable salts, derivatives and fragments, in which substitutes assume values given in the description.

EFFECT: compounds and pharmaceutical compositions containing said compounds can be used to treat diseases which are modulated by neuropeptide-2 receptors, mainly obesity.

13 cl, 10 dwg, 1 tbl, 74 ex

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RU 2 383 553 C2

Authors

Dankho Uolid

Ehrlich Dzhordzh

Fraj Dejvid S.

Kkhan Vadzhikha

Suistok Dzhozef

Dates

2010-03-10—Published

2006-01-11—Filed