COMBINATIONS CONTAINING ANTIMUSCARINE AGENTS AND CORTICOSTEROIDS Russian patent published in 2010 - IPC A61K31/439 A61K31/58 A61K31/573 A61P11/08 A61P11/06 

Abstract RU 2385156 C2

FIELD: medicine.

SUBSTANCE: invention covers drugs and concerns a combination intended for treating respiratory disease, containing (a) effective amount of corticosteroid, and (b) effective amount of antagonist of muscarine receptors M3 representing (3R)-1-phenethyl-3-(9N-xantene-9-xarbonyloxy)-1-azoniumbicyclo[2.2.2]octane in the form of salt with an anion X which represents a pharmaceutically acceptable anion of mono- or polyvalent acid. There is also disclosed application of (3R)-1-phenethyl-3-(9N-xantene-9-carbonyloxy)-1-azoniumbicyclo[2.2.2]octane and corticosteroid for making a drug for respiratory disease and the method of treating respiratory disease.

EFFECT: improved therapeutic effect in treating respiratory diseases.

20 cl, 1 dwg, 1 tbl, 7 ex

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RU 2 385 156 C2

Authors

Gras Ehskardo Khordi

L'Enas Kal'Vo Khesus

Rajder Khamish

Orvis Dias Pio

Dates

2010-03-27Published

2005-05-31Filed