FIELD: medicine.
SUBSTANCE: invention concerns to a derivative of formulas (I) and to its application as an inhibitor of human sodium-dependent glucose transporter (SGLT) for treating the diseases associated with hyperglycemia: 
, where A1 is O or S; A2 is CH or N; R1 or R4 is a group of formula (S): 
, where R5, R6 are hydrogen, hydroxyl, halogen, alkyl, alkoxy-, alkylthio; Q is alkylene, alkenylene, alkylene-O- alkylen-S-, -O-alkylene-, -S-alkylene-, alkylene-O-alkylene, -alkylene-S-alkylene-; A is phenyl; R2, R3 - hydrogen; G is group of formulae: 
or 
E1 - hydrogen, fluorine, hydroxyl; E2 - hydrogen, fluorine, methyl, hydroxymethyl.
EFFECT: production of new inhibitors of human SGLT.
15 cl, 17 ex, 7 tbl
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