ORGANIC COMPOUNDS Russian patent published in 2010 - IPC C07D498/22 A61K31/55 

Abstract RU 2394038 C2

FIELD: medicine.

SUBSTANCE: new crystal form II N-benzoilstaurosporin is described, as well as pharmaceutical composition containing it, inhibiting protein kinase C; ways of obtaining crystalline form of compounds, and the use of crystal form of II N-benzoilstaurosporin for treatment neoplastic diseases. Crystalline form of II N-benzoilstaurosporin is a stable form of N-benzoilstaurosporin with low hygroscopicity.

EFFECT: suitability in pharmaceutical compositions.

21 cl, 2 tbl, 4 dwg, 16 ex

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RU 2 394 038 C2

Authors

Ehn Paskal'

Kokh Bernd

Mutts Mikhaehl'

Dates

2010-07-10Published

2005-11-03Filed