CRYSTALLINE FORM III AND IV OF N-BENZOYLSTAUROSPORINE Russian patent published in 2016 - IPC C07D498/22 A61K31/553 A61P35/00 

Abstract RU 2598378 C2

FIELD: pharmaceutics.

SUBSTANCE: invention relates to a crystalline form III and a crystalline form IV of N-benzoyl staurosporine (midostaurin), pharmaceutical compositions based thereon.

EFFECT: treatment of leukemia, acute lymphoblastic leukaemia, myelodysplastic syndromes and mastocytosis; preparing pharmaceutical composition by extrusion of melt.

6 cl, 2 tbl, 4 dwg, 2 ex

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RU 2 598 378 C2

Authors

Randzhit Tkhakur

Dates

2016-09-27Published

2010-11-29Filed