CHEMICAL LINKERS AND CONJUGATES THEREOF Russian patent published in 2010 - IPC C07D403/14 C07D405/14 C07D417/14 A61K31/40 A61K49/18 A61K49/06 A61P35/00 

Abstract RU 2402548 C2

FIELD: chemistry.

SUBSTANCE: medicine-ligand conjugates are powerful cytotoxins in which the medicine is bonded to the ligand through a peptide, hydrazine or disulphide linker.

EFFECT: agents are highly effective.

63 cl, 8 ex

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Authors

Bojd Sharon

Chehn' Ljan

Gangvar Sandzhiv

Gerlaveh Vinsen

Khorgan Kilian

Li Chzhi-Khun

Sufi Bilal

Dates

2010-10-27Published

2005-05-19Filed