(S)-(-)-AMLODIPINE CAMSYLATE OR ITS HYDRATE AND PHARMACEUTICAL COMPOSITION INCLUDING THEM Russian patent published in 2010 - IPC C07D211/90 C07C309/07 A61K31/4422 A61P9/00 

Abstract RU 2403241 C1

FIELD: medicine, pharmaceutics.

SUBSTANCE: claimed invention relates to (S)-(-)-amlodipine camsylate of formula , where camphorsulfonic acid represents (1S)-(+)-10- camphorsulfonic acid or (±)-10- camphorsulfonic acid, as well as to its hydrate and to pharmaceutical composition, including them, which can be applied in treatment of cardiovascular diseases.

EFFECT: high photostability and solubility.

8 cl, 3 ex, 5 tbl, 4 dwg

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RU 2 403 241 C1

Authors

Li Dzaekheon

Li Moon Sub

Jang Veon Ki

Joo Dzaekho

Li Dzae-Chul

Choi Chang-Dzu

Kim Khan Kiong

Chang Jang-Kil

Li Gvansun

Dates

2010-11-10Published

2007-07-16Filed