COMPOUNDS, ENHANCING GLUTAMATE RECEPTOR, AND THEIR APPLICATION IN MEDICINE Russian patent published in 2010 - IPC C07D213/61 C07D239/26 C07D333/20 C07D213/42 C07D213/84 C07D237/08 C07D231/12 A61K31/44 A61K31/505 A61K31/381 A61K31/415 A61K31/4164 A61P25/08 

Abstract RU 2403242 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: claimed invention relates to compound of general formula (I) or its pharmaceutically acceptable salt, mediated by glutamate receptor, and to based on them pharmaceutical composition. (I), where R1 stands for C1-6alkyl; R2 and R3 stand for hydrogen; p stands for 0; n stands for 1; R5 and R6 stand for hydrogen, and Het stand for thienyl, pyridyl, pyrimidinyl, pyridazinyl, pyrazinyl, pyrazolyl, imidozolyl, each of which can be substituted with one or two groups, independently selected from the list, which consists of C1-6alkyl, C1-6alkoxy, acetyl, halogen, halogenC1-6alkyl, cyano.

EFFECT: creation of compound which has property to enhance response reaction.

4 cl, 2 tbl, 6 dwg, 38 ex

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RU 2 403 242 C2

Authors

Brehdli Dehniel Markus

T'Juliz Kevin Majkl

Uord Sajmon Ehdvard

Dates

2010-11-10Published

2005-08-05Filed