MICROPARTICLES CONTAINING ANALOGS OF SOMATOSTATIN Russian patent published in 2010 - IPC A61K9/16 A61K38/31 

Abstract RU 2404749 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention relates to pharmacology and medicine. Invention describes microparticles, including cyclo[{4-(NH2-C2H4-NH-CO-O-)Pro}-Phg-DTrp-Lys-Tyr(4-Bzl)-Phe] in free form, submerged into bio-compatible pharmacologically acceptable polymer matrix, where polymer matrix contains at least two different polymers selected from the group including linear and branched polylactide-co-glycolide for continuous release, and pharmaceutical compositions, including such microparticles.

EFFECT: production of pharmaceutical compositions, including microparticles - analogs of somatostatin.

13 cl, 11 ex, 4 tbl

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RU 2 404 749 C2

Authors

Al'Khajm Markus

Ausborn Mikhaehl'

Lamber Oliv'E

Rimenshnitter Mark

Dates

2010-11-27Published

2004-11-12Filed