N, N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS EFFECTIVE AS MONOAMINE REABSORPTION INHIBITORS Russian patent published in 2011 - IPC C07D207/14 C07D401/12 C07D401/14 C07D403/14 C07D405/12 C07D409/12 C07D413/12 C07D413/14 C07D417/12 C07D417/14 A61P25/00 

Abstract RU 2414454 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to new pyrrolidine derivatives of general formula (1) or its pharmaceutically acceptable salts where R101 and R102 values are described by the patent claim. The compounds inhibit serotonin and/or norepinephrine and/or dopamine reabsorption thereby allowing to be used for treating depression and anxiety disorder. A method for preparing thereof is described.

EFFECT: preparation of new pyrrolidine derivatives.

10 cl, 162 tbl, 7 ex

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RU 2 414 454 C2

Authors

Kurimura Muneaki

Taira Siniti

Tomojasu Takakhiro

Ito Nobuaki

Tai Kuninori

Takemura Noriaki

Matsuzaki Takajuki

Mendzo Jasukhiro

Mijamura Sin

Sakuraj Jokhdzi

Vatanabe Akikhito

Sakata Jasujo

Masumoto Takumi

Akazava Kokhej

Sugino Kharukhiko

Amada Naoki

Okhasi Satosi

Sinokhara Tomoiti

Sasaki Khirofumi

Morita Tisako

Jamasita Dzunko

Nakadzima Satoko

Dates

2011-03-20Published

2006-05-12Filed