FIELD: chemistry.
SUBSTANCE: invention relates to novel 5,7-diamino-substituted pyrazolo[1,5-a]pyrimidines selected from specific compounds, e.g. those given below, which have cyclin-dependent kinase inhibiting properties, such as CDK2. The compounds can be used to treat diseases and conditions associated with CDK, such as proliferative diseases, leukaemia.
.
EFFECT: more effective use of the compounds.
12 cl, 87 tbl, 1057 ex
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Authors
Dates
2011-03-20—Published
2005-02-08—Filed