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2 415 845

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IPC

C07D271/06(2006-01-01)

A61K31/4245(2006-01-01)

A61P31/06(2006-01-01)

A61P31/08(2006-01-01)

(21) (22)

Application

2009138082/04, 2009-10-14

(24)

Start date

2009-10-14

(22)

Actual filing date

2009-10-14

(45)

Published

2011-04-10

(72)

Inventor

Tyrkov Aleksej GeorgievichUrljapova Nelja GajfulovnaTyrkova Ekaterina Alekseevna

(73)

Holder

Gosudarstvennoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Gosudarstvennyj Universitet"

SULPHONIC 2-NITRO-2-(3-ARYL-1,2,4-OXADIAZOLE-5-YL)ETHANE DERIVATIVES EXHIBITING ANTILEPROTIC AND ANTITUBERCULOUS ACTIVITY Russian patent published in 2011 - IPC C07D271/06 A61K31/4245 A61P31/06 A61P31/08

Abstract RU 2415845 C1

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to sulphonic 2-nitro-2-(3-aryl-1,2,4-oxadiazole-5-yl)ethane derivatives of formula I a-g la R=3-NO₂C₆H4, R¹=NO₂, R²=H; b R=3-NO₂C₆H₄, R¹=NO₂, R²=CH₃; c R=4-CH₃OC₆H₄, R¹=NO₂, R²=H; d R=4-CH₃OC₆H₄, R¹=NO₂, R²=CH₃; e R=4-CH₃OC₆H₄, R¹=CO₂Et, R²=H; f R=4-CH₃OC₆H₄, R¹=CO₂Et, R²=CH₃; g R=4-CH₃C₆H₄, R¹⁼CO₂Et, R²=H.

EFFECT: preparation of the compound exhibiting antileprous and antituberculous activity.

1 cl, 1 tbl, 1 ex

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RU 2 415 845 C1

Authors

Tyrkov Aleksej Georgievich

Urljapova Nelja Gajfulovna

Tyrkova Ekaterina Alekseevna

Dates

2011-04-10—Published

2009-10-14—Filed