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2 420 521

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IPC

C07D271/06(2006-01-01)

C07D413/06(2006-01-01)

A61K31/4245(2006-01-01)

(21) (22)

Application

2009148583/04, 2009-12-25

(24)

Start date

2009-12-25

(22)

Actual filing date

2009-12-25

(45)

Published

2011-06-10

(72)

Inventor

Tyrkov Aleksej GeorgievichNosachev Svjatoslav BorisovichTjurenkov Ivan NikolaevichTimchenko Marija Vladimirovna

(73)

Holder

Gosudarstvennoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Gosudarstvennyj Universitet"

APPLICATION OF 1-HETARYL-2-NITRO-2-(3-PHENYL-1,2,4-OXADIAZOLE-5-YL)ETHANES AS PSYCHOTROPIC SUBSTANCES Russian patent published in 2011 - IPC C07D271/06 C07D413/06 A61K31/4245

Abstract RU 2420521 C1

FIELD: medicine.

SUBSTANCE: there is described application of 1-hetaryl-2-nitro-2-(3-phenyl-1,2,4-oxadiazole-5-yl)ethanes of general formula I a-m 1a, e, and R¹=NO₂, R²=H; 1b, f, to R¹=NO₂, R²=Me; 1c, g, l R¹=CO₂Et, R²=H; 1d, h, m R¹ =CO₂Et, R² =Me; 1a-d R² =piperidino; 1e-h R³ =1-pyrrolidinyl, 1j-m R³=morpholino as psychotropic substances.

EFFECT: substances are low-toxic and have an evident psychotropic effect on rats.

4 tbl, 4 ex

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RU 2 420 521 C1

Authors

Tyrkov Aleksej Georgievich

Nosachev Svjatoslav Borisovich

Tjurenkov Ivan Nikolaevich

Timchenko Marija Vladimirovna

Dates

2011-06-10—Published

2009-12-25—Filed