HYDROCHLORIDE SALT OF 5-[3-(3-HYDROXYPHENOXY)AZETIDIN-1-YL]-5-METHYL-2,2-DIPHENYLHEXANAMIDE Russian patent published in 2011 - IPC C07D205/04 A61K31/397 A61P11/00

Abstract RU 2422439 C2

FIELD: chemistry.

SUBSTANCE: invention also relates to a non-solvated crystalline form of the hydrochloride salt of 5-[3-(3-hydroxyphenoxy)azetidin-1-yl]-5-methyl-2,2-diphenylhexanamide, a pharmaceutical composition, use of compounds in claim 1 or 2, as well as a method of treating a mammal with M3 antagonist.

EFFECT: obtaining novel biologically active compounds which have M3 antagonist activity.

9 cl, 6 ex, 1 tbl

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RU 2 422 439 C2

Authors

Glossop Pol Alan

Dzhejms Kim

Dates

2011-06-27—Published

2008-03-06—Filed