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2 423 355

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IPC

C07D235/14(2006-01-01)

A61K31/4184(2006-01-01)

A61P31/04(2006-01-01)

(21) (22)

Application

2009134924/04, 2009-09-17

(24)

Start date

2009-09-17

(22)

Actual filing date

2009-09-17

(45)

Published

2011-07-10

(72)

Inventor

Morkovnik Anatolij Savel'EvichDivaeva Ljudmila NikolaevnaZubenko Aleksandr AleksandrovichPodladchikova Ol'Ga NikolaevnaFetisov Leonid NikolaevichAkopova Arina Romanovna

(73)

Holder

Federal'Noe Gosudarstvennoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Federal'Nyj Universitet" Ministerstva Nauki I Obrazovanija Rossijskoj Federatsii, Federal'Nogo Agentstva Po ObrazovanijuGosudarstvennoe Nauchnoe Uchrezhdenie Severo-Kavkazskij Zonal'Nyj Nauchno-Issledovatel'Skij Veterinarnyj Institut Rossijskoj Akademii Sel'Skokhozjajstvennykh Nauk

1,3-DISUBSTITUTED 2-IMINOBENZIMIDAZOLINE EXHIBITING ANTIBACTERIAL ACTION Russian patent published in 2011 - IPC C07D235/14 A61K31/4184 A61P31/04

Abstract RU 2423355 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: present invention refers to new benzimidazole derivatives of general formula I and to their pharmacologically acceptable salts, where lb R = CI, R¹ = H, R² = 3,4-Cl₂-C₆H₃; Ic R = H, R¹ = CH₃, R² = 3,4-C1₂-C₆H₃; Id R = H, R¹ = CI, R² = CONH₂; X = Cl^-, Br^-, showing antibacterial action.

EFFECT: new benzimidazole derivatives exhibiting high antibacterial activity are produced.

1 cl, 1 tbl

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RU 2 423 355 C2

Authors

Morkovnik Anatolij Savel'Evich

Divaeva Ljudmila Nikolaevna

Zubenko Aleksandr Aleksandrovich

Podladchikova Ol'Ga Nikolaevna

Fetisov Leonid Nikolaevich

Akopova Arina Romanovna

Dates

2011-07-10—Published

2009-09-17—Filed