FIELD: pharmacology.
SUBSTANCE: invention relates to the new derivatives in the 2,3,4,5-tetrahydro[1,3]diazepino [1,2-a]benzimidazole, with general formula 1:
.
The new hydrobromides 11-(4-t-butylbenzyl) - and 11-phenacyl substituted 2,3,4,5-tetrahydro[1,3]diazepino[1,2-A]benzimidazoles with anxiolytic activity are obtained.
EFFECT: improved compounds properties.
4 cl, 2 tbl, 3 ex
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