SUCCINATE OF N-(2,4,6-TRIMETHYLPHENYL)AMIDE 2-(BETA-N,N-DIETHYLAMINO ETHYLAMINO)-4-OXO-4-(4-METHYYLPHENYL)-2-BUTENOIC ACID Russian patent published in 2011 - IPC C07C237/20 A61P23/02 A61K31/167 

Abstract RU 2428412 C2

FIELD: chemistry.

SUBSTANCE: novel compound relates to amine derivatives of pyruvic acid amides and is biologically active - succinate of N-(2,4,6-trimethylphenyl) amide 2-(β-N,N-diethylamino ethylamino)-4-oxo-4-(4-methyl-phenyl)-2-butenoic acid of formula

.

EFFECT: compound has marked local anaesthetic and antimicrobial activity.

1 cl, 1 ex, 3 tbl

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Authors

Borodin Anton Jur'Evich

Igidov Nazim Musabekovich

Mel'Nikova Natal'Ja Aleksandrovna

Chashchina Svetlana Viktorovna

Odegova Tat'Jana Fedorovna

Borodina Tat'Jana Viktorovna

Dates

2011-09-10Published

2009-10-15Filed