FIELD: medicine, pharmaceutics.
SUBSTANCE: invention refers to pharmaceutical chemistry, more specifically to a method for producing octreotide by a liquid phase method by oxidative ring formation with using potassium triiodide in a water-methanol solution as an oxidative and unblocking reagent.
EFFECT: method is characterised by simplicity, absence of toxic reagents and high yield of an end product.
2 ex
Title | Year | Author | Number |
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PROTECTED DERIVATIVES OF OCTREOTIDE | 2001 |
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Authors
Dates
2011-12-10—Published
2010-07-08—Filed