THERAPEUTIC ANTIDIABETIC AGENT Russian patent published in 2012 - IPC A61K31/506 A61K31/54 A61P1/18 A61P3/10 

Abstract RU 2438671 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: present invention refers to pharmaceutics and medicine, and concerns a pancreas protector which contains a combination of a blood glucose decreasing drug not stimulating insulin secretion and a compound presented by formula (1), where the compound of formula (1) represents 2-[[6-[(3R)-3-amino-1-piperidinyl]-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl]methyl]benzonitrile or 2-[[6-[(3R)-3-amino-1-piperidinyl]-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl]methyl]-4-fluorobenzonitrile exhibiting higher efficacy.

EFFECT: improved efficacy of the preparation.

15 cl, 4 tbl, 4 ex

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RU 2 438 671 C2

Authors

Takeuti Kodzi

Moritokh Jusuke

Dates

2012-01-10Published

2006-12-27Filed