FIELD: medicine, pharmaceutics.
SUBSTANCE: declared invention refers to chemical-pharmaceutical industry, and concerns 2,2,2-Trifluoro-1-trifluoromethylethyl ester of cyclohexylcarbamine acid 
which is prepared starting with cyclohexylisocyanate and 1-hydrohexafluorisopropanole at 20°C in benzene in the presence of catalytic amounts of triethylamine.
EFFECT: compound (I) is an effective and selective irreversible carboxylesterase inhibitor with low acute toxicity in warm-blooded, and may be used in preclinical studies on rodents for decreasing carboxylesterase hydrolysis rate of the drugs containing ester and/or amide groups, and also as insect carboxylesterase inhibitors in pharmaceutical composition and pesticide formulations for increasing their efficacy.
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