SOLID FORMS OF RACEMIC ILAPRAZOLE Russian patent published in 2012 - IPC C07D401/14 A61K31/4439 A61P1/04 

Abstract RU 2466129 C2

FIELD: chemistry.

SUBSTANCE: present invention relates to crystalline forms A, B and F of racemic ilaprazole (2[[(4-methoxy-3-methyl-2-pyridinyl)-methyl]thionyl]-5-(1H-pyrrol-1-yl)-1H-benzimidazole). The invention also relates to a pharmaceutical composition based on crystalline ilaprazole and use of crystalline ilaprazole.

EFFECT: obtaining novel crystalline forms of ilaprazole which can be used to inhibit gastric acid secretion.

14 cl, 57 dwg, 39 tbl, 10 ex

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RU 2 466 129 C2

Authors

Brakett Dzhon M.

Dzhonajtis Dehvid T.

Laj Vej

L'Ju Dzhikh Khua

Parent Stefan D.

Shen Dzhinuju

Dates

2012-11-10Published

2007-12-28Filed