N-[3-OXO-LUPANO-28-YL]-PIPERIDINE - AGENT HAVING ANTI-TUMOUR, ANTI-METASTATIC, ANTI-INFLAMMATORY AND CYTOPROTECTIVE ACTIVITY Russian patent published in 2012 - IPC C07J43/00 C07J53/00 A61P35/00 

Abstract RU 2466136 C1

FIELD: chemistry.

SUBSTANCE: invention relates to a novel chemical compound and specifically to N-[3-oxo-lupano-28-yl]-piperidine of formula (1): having complex activity - anti-tumour, anti-metastatic, anti-inflammatory and cytoprotective activity. The compound is synthesised from dihydrobetulonic acid.

EFFECT: obtaining compounds for reducing proliferation and dissemination of malignant cells and relieving necrobiotic disorders in normal cells, arising under the influence of paraneoplastic processes and cytotoxic chemotherapy.

1 cl, 11 ex, 7 tbl, 4 dwg

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RU 2 466 136 C1

Authors

Sorokina Irina Vasil'Evna

Tolstikova Tat'Jana Genrikhovna

Zhukova Tat'Jana Anatol'Evna

Bessergeneva Ekaterina Pavlovna

Majnagashev Il'Ja Jakovlevich

Salakhutdinov Nariman Faridovich

Tolstikov Genrikh Aleksandrovich

Dates

2012-11-10Published

2011-07-19Filed