PHOSPHONIUM SALTS ON BASIS OF PYRIDOXINE DERIVATIVES Russian patent published in 2012 - IPC A61K31/66 C07F9/54 C07D213/67 

Abstract RU 2466728 C1

FIELD: medicine.

SUBSTANCE: invention refers to phosphonium salt of pyridoxine derivatives of general formula (I) which may be used in medicine and veterinary science wherein if R1=CH3; R2=CH3; X=H; n=1; R1=CH3; R2=H; X-H; n=1; R1=CH3; R2=CH3; X-CH2P*Ph3; n=2; R,=CH3; R2=H; X=CH2P+Ph3; n=2; R,=CH3; R2=C(CH3)2; X=CH2P+Ph3; n=2.

EFFECT: there are presented new compounds with antibacterial activity on Staphylococcus aureus, including multiresistant strains, as well as low toxicity.

1 cl, 1 ex, 1 tbl

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RU 2 466 728 C1

Authors

Shtyrlin Jurij Grigor'Evich

Shtyrlin Nikita Valer'Evich

Pugachev Mikhail Vladimirovich

Dates

2012-11-20Published

2011-09-12Filed