FIELD: chemistry.
SUBSTANCE: invention relates to biologically active compounds, specifically to a group of 2-substituted 1,2,4,5-tetrahydro-3H-pyrrolo[1,2-a][1,4]diazepin-3-ones of general formula 
where R denotes hydrogen, a straight or branched (C1-C4)-alkyl; a hydroxyalkyl having an alkyl chain with 2-3 C atoms; a phenylalkyl having an alkyl chain with 1-2 C atoms, wherein the phenyl ring can have one or two methoxy groups. The invention also relates to a method of producing said compounds.
EFFECT: novel compounds can be used in medicine as antidepressant and antianxiety agents.
6 cl, 3 tbl, 9 ex
| Title | Year | Author | Number |
|---|---|---|---|
| USE OF 5-(4-METOXYPHENYL)-7-METHYL-1,2,4,5-TETRAHYDRO-3H-PYRROLO[1,2-a][1,4]DIAZEPIN-3-ONE AS AN ANTIFUNGAL AGENT AGAINST YEAST FUNGI | 2023 |
|
RU2810715C1 |
| USE OF 7-METHYL-5-[4-(TRIFLUOROMETHYL)PHENYL]-1,2,4,5-TETRAHYDRO-3H-PYRROLO[1,2-a][1,4]DIAZEPIN-3-ONE AS AN ANTIFUNGAL AGENT AGAINST YEAST FUNGI | 2023 |
|
RU2808981C1 |
| USE OF 2-METHYL-4-[7-(TRIFLUOROMETHYL)PHENYL]-1,2,4,5-TETRAHYDRO-3H-PYRROLO[1,2-a][1,4]DIAZEPIN-3-ONE AS ANTIFUNGAL AGENT AGAINST YEAST FUNGI | 2023 |
|
RU2809051C1 |
| USE OF 7-METHYL-2-(4-METHYLPHENYL)-1,2,4,5-TETRAHYDRO-3H-PYRROLO[1,2-a][1,4]DIAZEPIN-3-ONE AS AN ANTIFUNGAL AGENT AGAINST YEAST FUNGI | 2023 |
|
RU2809053C1 |
| 1-ARYLPYRROLO[1,2A]PYRAZINE-3-CARBOXAMIDES WITH NEUROPSYCHOTROPIC ACTIVITY | 2014 |
|
RU2572076C2 |
| METHOD FOR PRODUCTION OF 4-ARYL-2,7,9-TRIAZASPIRO[4,5]DECANE-6,8,10-TRIONS | 2016 |
|
RU2635105C1 |
| PYRAZOLE DERIVATIVES APPLIED AS PROTEIN KINASE INHIBITORS | 2013 |
|
RU2623221C2 |
| METHOD FOR PRODUCING OF 7-ALKYL-2,3-DIHYDRO-1H-PYRROLO[1,2-D][1,4]DYAZEPINE-4(5H)-ONE DERIVATIVES | 2017 |
|
RU2659390C1 |
| METHOD OF PRODUCING 5,6-DIHYDRO-4H-BENZO[f]PYRROLO[1,2-α][1,4]DIAZEPIN-6-ONE | 2010 |
|
RU2425037C1 |
| NOVEL PHOSPHATE COMPOUNDS, SYNTHESIS METHOD THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME | 2014 |
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RU2617682C2 |
