FIELD: chemistry.
SUBSTANCE: invention relates to a folate receptor ligand which is folate-polyethylene glycol-dihexadecyl-L-glutamate of formula 
and a method for production thereof. This compound exhibits the capacity to direct a nanosystem to target cells and increases the efficiency of transportation systems of antitumour agents since folate receptors are present in large amounts on the surface of tumour cells; also they become more at the later stages of development of the disease.
EFFECT: use of an approach based on click-chemistry principles for synthesis of a folate-targeted derivative provides a unique opportunity for fast and efficient modification of nanosystems.
2 cl
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