STABILISED PHARMACEUTICAL DOCETAXEL-CONTAINING COMPOSITION Russian patent published in 2013 - IPC A61K9/08 A61K31/337 A61K47/08 A61P35/00 

Abstract RU 2478370 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: claimed invention relates to medicine and describes pharmaceutical composition for injecting, based on homogeneous liquid, containing docetaxel, with controlled pH in the interval from 3 to 5, consisting of: (a) docetaxel or its pharmaceutically acceptable salt, (b) surfactant, selected from group, consisting of polysorbate, polyoxyethylene glycol ester and polyoxyethylene derivatives of castor oil, (c) water-free ethanol in concentration from 100 to 800 mg/ml, and (d) pH regulator, selected from citric acid, fumaric acid, lactic acid, stannic acid, succinic acid, maleic acid, acetic acid, tartaric acid and phosphoric acid.

EFFECT: composition is suitable for efficient introduction of docetaxel as it has improved pharmaceutical stability.

2 cl, 4 ex, 8 tbl

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RU 2 478 370 C2

Authors

Ju Mu-Khi

Cha Bon-Chzhin

Kim Chzhon-Khun

Chan Sun-Vu

Von Don-Khan

Dates

2013-04-10Published

2009-02-26Filed