INTERMEDIATE COMPOUNDS AND METHODS FOR PREPARING ZEARALENE MACROLIDE ANALOGUES Russian patent published in 2013 - IPC C07D313/00 C07C69/66 C07D491/04 

Abstract RU 2478630 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: present invention refers to methods for preparing macrolides, e.g. compounds of formula (IV) and intermediate compounds of formula (V):

and , wherein R1-R12 have the values specified in the description.

EFFECT: compounds of formula V are valuable for treating inflammatory or immune disorders, and treating cancer.

12 cl, 12 dwg, 18 ex

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Authors

Buaven Rosh

Kampan'Ja Sil'Vio A.

Du Khun

Fan Frehnsis Dzh.

Khorstmann Tomas

Lemelin Sharl'-Andre

Li Tszin

Maksginness Pamela

Nju Sjan

Shnaderbek Mehtt'Ju Dzh.

U Kevin

Chzhu Sjaotsze

Dates

2013-04-10Published

2008-12-08Filed