19-NOR C3,3-DISUBSTITUTED C21-N-PYRAZOLYL STEROIDS AND METHODS OF THEIR USE Russian patent published in 2024 - IPC C07J7/00 C07J43/00 A61K31/58 A61P25/00 

Abstract RU 2812930 C2

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to the use of a compound of the formula:

for treating one or several of the following GABA-mediated disorders: mood disorder, anxiety disorder, bipolar disorder, tremor or tinnitus in a subject in need thereof and for inhibiting or potentiating GABA receptor function in a subject suffering from one or several of the following GABA-mediated disorders: affective disorder, anxiety disorder, bipolar disorder, tremors or tinnitus.

EFFECT: obtaining of a new compound that is active against the GABA receptor and can be used to treat an indirect disorder.

27 cl, 5 tbl, 52 dwg, 71 ex

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RU 2 812 930 C2

Authors

Botella, Gabriel Martinez

Harrison, Boyd L.

Robichaud, Albert Jean

Salituro, Francesco G.

Beresis, Richard Thomas

Dates

2024-02-05Published

2014-04-17Filed