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2 539 595

(13)

(51)

IPC

C07D261/04(2006-01-01)

C07D413/04(2006-01-01)

C07D413/12(2006-01-01)

C07D413/14(2006-01-01)

C07D498/04(2006-01-01)

C07D498/10(2006-01-01)

A61K31/42(2006-01-01)

A61P29/00(2006-01-01)

A61P37/02(2006-01-01)

A61P25/00(2006-01-01)

(21) (22)

Application

2011151635/04, 2010-05-18

(24)

Start date

2010-05-18

(22)

Actual filing date

2010-05-18

(45)

Published

2015-01-20

(72)

Inventor

Benke Mark L.Kastro Al'Fredo S.Chan Lourens K.Ehvans Kehtrin A.Gren'E LuiGrogan Majkl Dzh.Leblan IvLju TaoPeljuzo StefanSnajder Dehniel A.Tibbitts Tomas T.

(73)

Holder

Infiniti Farmas'Jutikalz, Ink.

ISOXAZOLINE AS FATTY ACID AMIDE HYDROLASE INHIBITORS Russian patent published in 2015 - IPC C07D261/04 C07D413/04 C07D413/12 C07D413/14 C07D498/04 C07D498/10 A61K31/42 A61P29/00 A61P37/02 A61P25/00

Abstract RU 2539595 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: present invention refers to isoxazoline FAAH inhibitors of formula (I) or their pharmaceutically acceptable forms, wherein each of G, R^a, R^b, R^c and R^d has a value described in the present application, to pharmaceutical compositions, and methods of treating a FAAH-mediated condition.

EFFECT: developing the method of treating the FAAH-mediated condition.

32 cl, 22 tbl, 351 ex

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RU 2 539 595 C2

Authors

Benke Mark L.

Kastro Al'Fredo S.

Chan Lourens K.

Ehvans Kehtrin A.

Gren'E Lui

Grogan Majkl Dzh.

Leblan Iv

Lju Tao

Peljuzo Stefan

Snajder Dehniel A.

Tibbitts Tomas T.

Dates

2015-01-20—Published

2010-05-18—Filed