FIELD: medicine, pharmaceutics.
SUBSTANCE: there are described new 1,2,4-triazine-3,5-dione derivatives of general formula 
(I) wherein A is a saturated hydrocarbon chain with chain length 4 to 6 atoms; R1 and R2 are optionally hydrogen or C1-C3-alkyl; R3 is branched C4-C6-alkyl or C3-C6-cycloalkyl; R4 - C1-C6-alkyl, C3-C6-cycloalkyl or fluorinated C1-C3-alkyl, their physiologically acceptable salts and N-oxides, and a pharmaceutical composition containing them.
EFFECT: new compounds show dopamine D3 receptor activity and may be used in treating the central nervous system diseases.
24 cl, 8 ex, 1 tbl
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