FIELD: medicine, pharmaceutics.
SUBSTANCE: invention refers to tetraazaphenalen-3-one compounds, particularly a compound of formula 
which inhibit poly(ADP-ribose)polymerase (PARP) and may be used for chemosensitisation in relation to anticancer chemotherapeutic agents.
EFFECT: higher effectiveness of the chemotherapeutic agents, and in treating cancer diseases characterised by the DNA repair defects.
13 cl, 2 tbl, 6 dwg, 3 ex
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