THIAZOLIDINEDIONE ANALOGUES FOR TREATING DIABETES AND DYSLIPIDEMIA Russian patent published in 2013 - IPC C07D277/34 A61K31/426 A61P9/12 A61P3/10 A61P29/00 

Abstract RU 2486179 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to a selective thiazolidinedione analogue to be used in treating and preventing diabetes and dyslipidemia, representing 5-(4-(2-(3-methoxyphenyl)-2-oxoethoxy)benzyl)thiazolidine-2,4-dione or a pharmaceutically acceptable salt thereof. Also, the invention refers to a pharmaceutical composition for diabetes and dyslipidemia, containing an effective amount of 5-(4-(2-(3-methoxyphenyl)-2-oxoethoxy)benzyl)thiazolidine-2,4-dione or the pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier. .

EFFECT: what is produced is the selective thiazolidinedione analogue decreasing binding and activating of the PPARγ nuclear transcription factor.

4 cl, 2 tbl, 10 ex

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RU 2 486 179 C2

Authors

Kolka Dzherard R.

Gehdvud Robert K.

Parker Tim

Dates

2013-06-27Published

2008-09-15Filed