METHOD FOR GLYCOSIDATION OF COLCHICINE AND THIOCOLCHICINE Russian patent published in 2013 - IPC C07H15/248 C07C49/755 

Abstract RU 2488589 C2

FIELD: chemistry.

SUBSTANCE: present invention discloses a method of producing compounds of formula I, wherein: R1 is a methoxy or methylthio group; R2 is an O-glycosyloxy residue. Compounds of formula I are obtained by reacting peracetylated glucose with a compound of formula II , followed by removal of protective groups from the glycosyl moiety.

EFFECT: high efficiency of the method.

9 cl, 4 ex

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RU 2 488 589 C2

Authors

Beszant Stefen

Gabetta Bruno

Dates

2013-07-27Published

2009-04-09Filed